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Sarpogrelate hydrochloride
CAS No. 135159-51-2
Sarpogrelate hydrochloride ( MCI 9042;MCI9042;MCI-9042 )
Catalog No. M11420 CAS No. 135159-51-2
A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 37 | In Stock |
|
| 10MG | 59 | In Stock |
|
| 25MG | 110 | In Stock |
|
| 50MG | 176 | In Stock |
|
| 100MG | 259 | In Stock |
|
| 500MG | 619 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSarpogrelate hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
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DescriptionA potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.Heart Failure Approved
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SynonymsMCI 9042;MCI9042;MCI-9042
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number135159-51-2
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Formula Weight465.97
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Molecular FormulaC24H32ClNO6
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 62 mg/mL
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SMILESCN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl
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Chemical NameButanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
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