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Sarpogrelate hydrochloride

CAS No. 135159-51-2

Sarpogrelate hydrochloride ( MCI 9042;MCI9042;MCI-9042 )

Catalog No. M11420 CAS No. 135159-51-2

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Sarpogrelate hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
  • Description
    A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.Heart Failure Approved
  • Synonyms
    MCI 9042;MCI9042;MCI-9042
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    135159-51-2
  • Formula Weight
    465.97
  • Molecular Formula
    C24H32ClNO6
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 62 mg/mL
  • SMILES
    CN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl
  • Chemical Name
    Butanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
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